M.Wt: 338.25
Formula: C14H12F6N2O - 4-((R)-2-((R)-2,2,2-trifluoro-1-hydroxyethyl)pyrrolidin-1-yl)-2-trifluoroMethyl)benzonitrile
Solubility: DMSO
Purity: >99%
Storage: at 20ºC 2 years
Half life: 24 hours
CAS No.: 1165910-22-4
ACTIVITY OF LGD-4033:
LGD-4033 is a selective androgen receptor modulator a novel non-steroidal, oral SARM that binds to AR with high affinity (Ki of ~1 nM) and selectivity, class of androgen receptor (AR) ligands that is tissue selective, developed to treat muscle wasting associated with cancer, acute and chronic illness and age-related muscle loss. Expected to produce the therapeutic benefits of testosterone with improved safety, tolerability and patient acceptance due to tissue-selective mechanism of action and an oral route of administration. It demonstrates anabolic activity in muscles, anti-resorptive and anabolic activity in bones and a robust selectivity for muscle and bone versus prostate and sebaceous glands. LGD-4033 has recently completed a Phase I Multiple Ascending Dose study in healthy volunteers this randomized, double-blind, placebo-controlled Phase I study established the safety and tolerability up to doses of 22 mg.
Certificate of Analysis |
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Product Name | LGD 4033 /Ligandrol |
Batch No | 180125 |
Quantity | 10kg | Produce Date | 2018.03.06 |
Ref Standard |
| Exp Date | 2019.03.07 |
Items And Results |
Item | Quality level | Determination |
Appearance | white powder | White powder |
HNMR | Conforms to structure | conforms |
LCMS | Conforms to MW | conforms |
Assay | ≥98.5% | 99.00% |
Conclusion | Passed |
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Packing description | Sealed export grade drum & double of sealed plastic bag |
Storage | Store in cool & dry place not freeze, keep away from strong light and heat |
Shelf life | 1 years when properly stored |
YK11 | 1370003-76-1 |
OSTARINE/MK2866 | 1202044-20-9 841205-47-8 1235370-13-4 |
GW501516/Cardarine | 317318-70-0 |
GW0742 | 317318-84-6 |
MK677 / Ibutamoren | 159752-10-0 |
AICAR | 2627-69-2 |
SR9009 | 1379686-30-2 |
SR9011 | 1379686-29-9 |
RAD 140 | 1182367-47-0 |
AC 262,356 | 870888-46-3 |
ACP 105 | 899821-23-9 |
LGD 4033 /Ligandrol | 1165910-22-4 |
LGD 3033 |
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Capromorelin | 193273-66-4 |
S4 | 401900-40-1 |
S-23 | 1010396-29-8 |